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EZM0414 TFA
CAS No. 2411759-92-5
EZM0414 TFA( —— )
Catalog No. M34899 CAS No. 2411759-92-5
EZM0414 TFA (SETD2-IN-1 TFA) is a SETD2 inhibitor with anticancer and antiproliferative effects for the study of leukemia and immune dysfunction.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 454 | Get Quote |
|
| 500MG | Get Quote | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NameEZM0414 TFA
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NoteResearch use only, not for human use.
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Brief DescriptionEZM0414 TFA (SETD2-IN-1 TFA) is a SETD2 inhibitor with anticancer and antiproliferative effects for the study of leukemia and immune dysfunction.
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DescriptionEZM0414 TFA is a potent, selective and orally active inhibitor of SETD2 which is a human histone methyltransferase. EZM0414 TFA has anti-proliferative effects.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayOthers
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TargetOther Targets
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RecptorHistone Methyltransferase
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Research Area——
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Indication——
Chemical Information
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CAS Number2411759-92-5
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Formula Weight514.51
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Molecular FormulaC24H30F4N4O4
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 200 mg/mL (388.72 mM; Ultrasonic ) H2O : 6.67 mg/mL (12.96 mM; Ultrasonic (<60°C))
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SMILESOC(=O)C(F)(F)F.CC(=O)N1CCN(CC1)[C@H]1CCC[C@H](C1)NC(=O)c1cc2c(F)ccc(C)c2[nH]1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. John Lampe, et al. Substituted indoles and methods of use thereof. WO2020037079A1.
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